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CRIZOTINIB
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DeCS
Descriptor
English
:
Crizotinib
Descriptor
Spanish
:
crizotinib
Descriptor
Portuguese
:
Crizotinibe
Synonyms
English
:
PF 02341066
PF 2341066
PF-02341066
PF-2341066
PF02341066
PF2341066
Xalkori
Tree Number:
D03.383.621.154
D03.383.725.050.263
Definition
English
:
A piperidine and aminopyridine derivative that acts as an inhibitor of
RECEPTOR PROTEIN-TYROSINE KINASES
, including
ANAPLASTIC LYMPHOMA KINASE
(ALK) and
HEPATOCYTE GROWTH FACTOR
RECEPTOR (HGFR; c-Met). It is used in the treatment of NON-SMALL CELL LUNG CANCER.
Pharmacological Action:
Antineoplastic Agents
Protein Kinase Inhibitors
History Note
English
:
2019 (2010)
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AA
analogs & derivatives
AN
analysis
AI
antagonists & inhibitors
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
57672
Unique Identifier:
D000077547
Occurrence in VHL
:
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