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COBICISTAT
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DeCS
Descriptor
English
:
Cobicistat
Descriptor
Spanish
:
cobicistat
Descriptor
Portuguese
:
Cobicistat
Synonyms
English
:
9350, GS
GS 9350
GS-9350
GS9350
Tybost
Tree Number:
D02.241.081.251.203
D02.886.675.182
D03.383.129.708.189
Definition
English
:
A carbamate and thiazole derivative that functions as a
CYTOCHROME
P450 CYP3A INHIBITOR to enhance the concentration of
ANTI-HIV AGENTS
, with which it is used in combination, for the treatment of
HIV INFECTIONS.
Pharmacological Action:
Anti-HIV Agents
Cytochrome P-450 CYP3A Inhibitors
History Note
English
:
2016 (2011)
Allowable Qualifiers
English
:
AD
administration & dosage
AE
adverse effects
AG
agonists
AA
analogs & derivatives
AN
analysis
AI
antagonists & inhibitors
BL
blood
CF
cerebrospinal fluid
CS
chemical synthesis
CH
chemistry
CL
classification
EC
economics
HI
history
IM
immunology
IP
isolation & purification
ME
metabolism
PK
pharmacokinetics
PD
pharmacology
PO
poisoning
RE
radiation effects
ST
standards
SD
supply & distribution
TU
therapeutic use
TO
toxicity
UR
urine
Record Number:
55886
Unique Identifier:
D000069547
Occurrence in VHL
:
Similar:
DeCS